SCHEMBL100288

SCHEMBL100288

O=C(O)Nc1cc(CCC(=O)Nc2ccc(CO)c(Cl)c2)ccc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.46
HCAR2 Q8TDS4 5/20 0.45
RORC P51449 1/20 0.45
MAPT P10636 3/20 0.43
GAA P10253 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL101227 0.95 NPC1 (0.45) PTGDR2HCAR2RORCMAPTMEN1
SCHEMBL100326 0.88 HCAR2 (0.46) HCAR2MAPTGAAAKR1C3AKR1C2
SCHEMBL100587 0.88 RORC (0.46) HCAR2RORCMAPTGAAAKR1C3
SCHEMBL98704 0.86 AKR1C3 (0.51) HCAR2RORCMAPTGAAAKR1C3
SCHEMBL99091 0.85 RAB9A (0.51) MAPTGAAMEN1KMT2ANPC1
SCHEMBL101812 0.84 PTGDR2 (0.42) PTGDR2HCAR2RORCMAPTNPC1
SCHEMBL99215 0.83 AKR1C3 (0.49) HCAR2MAPTGAAAKR1C3AKR1C2
SCHEMBL99701 0.82 AKR1C3 (0.53) HCAR2AKR1C3AKR1C2MEN1KMT2A
SCHEMBL101223 0.81 HDAC1 (0.51) MAPTAKR1C3AKR1C2MEN1KMT2A
SCHEMBL662760 0.81 CHRM3 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed