SCHEMBL10035933

SCHEMBL10035933

COc1cc(N)ccc1NC1CCN(C)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 9/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
HSD17B10 Q99714 1/20 0.49
EZH2 Q15910 2/20 0.46
DNMT1 P26358 1/20 0.46
EHMT1 Q9H9B1 5/20 0.46
QDPR P09417 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CDK1 P06493 1/20 0.43
POLB P06746 1/20 0.43
NSD2 O96028 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12988943 0.85 EHMT2 (0.49) EHMT2ALDH1A1GAAHSD17B10EZH2
SCHEMBL10808825 0.84 GAA (0.47) ALDH1A1GAAHSD17B10
SCHEMBL1814668 0.81 FLT3 (0.45) EHMT2ALDH1A1GAADNMT1POLB
SCHEMBL31203040 0.81 FLT3 (0.45) EHMT2ALDH1A1GAADNMT1POLB
SCHEMBL29972689 0.80 POLB (0.44) EHMT2ALDH1A1GAAPOLB
SCHEMBL3023350 0.80 POLB (0.44) EHMT2ALDH1A1GAAPOLB
SCHEMBL13459865 0.79 DRD2 (0.46) QDPR
SCHEMBL5257134 0.79 QDPR (0.44) GAAQDPRNSD2
SCHEMBL10035929 0.78 NPSR1 (0.56) ALDH1A1GAACYP3A4
SCHEMBL282999 0.77 QDPR (0.52) EHMT2GAAQDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053606-A1 ARYLAMINOHETEROCYCLIC CARBOXAMIDE COMPOUND アステラス製薬株式会社 (JP) 2012-04-26 WO disclosed