SCHEMBL10042987

SCHEMBL10042987

CC1=C(C)C(C(N)=O)C(NC(=O)CN(Cc2ccco2)C(=O)c2ccccc2)S1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
CYP2C19 P33261 3/20 0.48
LMNA P02545 3/20 0.48
MAPT P10636 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C9 P11712 2/20 0.48
HTT P42858 1/20 0.48
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 3/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.43
USP2 O75604 1/20 0.43
HSD17B10 Q99714 1/20 0.43
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10042833 0.84 ALDH1A1 (0.43) ALDH1A1LMNAHDAC1HDAC6NPSR1
SCHEMBL10042806 0.71 ALDH1A1 (0.63) ALDH1A1CYP2C19LMNAMAPTCYP1A2
SCHEMBL5641649 0.64 HPGD (0.58) ALDH1A1CYP2C19LMNAMAPTCYP1A2
SCHEMBL12900896 0.63 HDAC1 (0.68) MAPTHDAC1HDAC6POLB
SCHEMBL2834886 0.63 ALOX5 (0.56) ALDH1A1CYP2C19LMNAMAPTCYP1A2
SCHEMBL12900897 0.63 HDAC1 (0.60) ALDH1A1LMNAMAPTHDAC1HDAC6
SCHEMBL12934246 0.62 MAPT (0.77) ALDH1A1MAPTHDAC1HDAC6SMN1; SMN2
SCHEMBL12231378 0.61 ALDH1A1 (0.79) ALDH1A1CYP2C19LMNAMAPTCYP1A2
SCHEMBL30639187 0.61 SMN1; SMN2 (0.52) ALDH1A1CYP2C19LMNAMAPTCYP1A2
SCHEMBL29141346 0.61 SMN1; SMN2 (0.52) ALDH1A1CYP2C19LMNAMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018932-A2 COMPOUNDS AND COMPOSITIONS FOR MITIGATING TISSUE DAMAGE AND LETHALITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-02-09 WO disclosed