SCHEMBL10042833

SCHEMBL10042833

CC1=C(C)C(C(N)=O)C(NC(=O)CN(Cc2ccc(F)cc2)C(=O)c2ccccc2)S1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
CTSS P25774 4/20 0.43
CTSL P07711 2/20 0.43
CTSK P43235 2/20 0.42
AGER Q15109 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MTNR1A P48039 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HDAC1 Q13547 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10042987 0.84 ALDH1A1 (0.48) ALDH1A1LMNAMEN1KMT2ANPSR1
SCHEMBL10042805 0.71 LMNA (0.74) ALDH1A1LMNAMEN1KMT2ANPSR1
SCHEMBL16109738 0.66 HDAC1 (0.65) ALDH1A1MEN1KMT2ANPSR1HDAC1
SCHEMBL5645455 0.64 NSD2 (0.67) MEN1KMT2AHDAC1HDAC6
SCHEMBL12231196 0.63 LIMK2 (0.52) ALDH1A1LMNAMEN1KMT2ARAB9A
SCHEMBL29190232 0.62 HDAC1 (0.61) ALDH1A1LMNAMEN1KMT2AHDAC1
SCHEMBL569976 0.62 ALDH1A1 (0.82) ALDH1A1LMNACTSSCTSLMEN1
SCHEMBL1500765 0.61 BCL2 (0.60) ALDH1A1LMNAMEN1KMT2ANPSR1
SCHEMBL30482165 0.61 TDP1 (0.49) ALDH1A1LMNAAGERMEN1KMT2A
SCHEMBL3640312 0.61 HCRTR1 (0.57) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018932-A2 COMPOUNDS AND COMPOSITIONS FOR MITIGATING TISSUE DAMAGE AND LETHALITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-02-09 WO disclosed