SCHEMBL10046161

SCHEMBL10046161

Bc1cc(N)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
MAPK1 P28482 1/20 0.46
NR2E1 Q9Y466 1/20 0.39
KIF11 P52732 3/20 0.38
PTPN5 P54829 2/20 0.35
ALDH1A1 P00352 3/20 0.34
IDO1 P14902 2/20 0.34
MAPT P10636 1/20 0.34
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
PKM P14618 1/20 0.34
CES2 O00748 1/20 0.33
GLA P06280 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
IKBKB O14920 1/20 0.31
BACE1 P56817 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL394717 0.82 TSHR (0.56) TSHRMAPK1NR2E1KIF11PTPN5
SCHEMBL130383 0.82 TSHR (0.56) TSHRMAPK1NR2E1KIF11PTPN5
SCHEMBL19270461 0.82 CES2 (0.40) TSHRMAPK1PTPN5ALDH1A1IDO1
SCHEMBL3684529 0.82 CES2 (0.46) TSHRMAPK1ALDH1A1IDO1MAPT
SCHEMBL29136201 0.79 CES2 (0.44) TSHRMAPK1ALDH1A1IDO1MAPT
Iodide SCHEMBL31550893 0.79 TSHR (0.54) TSHRMAPK1NR2E1KIF11PTPN5
SCHEMBL28802521 0.79 CES2 (0.44) TSHRMAPK1ALDH1A1IDO1MAPT
SCHEMBL27859051 0.79 TSHR (0.54) TSHRMAPK1NR2E1KIF11PTPN5
Hydrochloric Acid SCHEMBL9741395 0.79 TSHR (0.54) TSHRMAPK1NR2E1KIF11PTPN5
Water SCHEMBL27788452 0.79 CES2 (0.44) TSHRMAPK1ALDH1A1IDO1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896426-B1 PROCESS FOR THE SYNTHESIS OF ORGANIC COMPOUNDS NOVARTIS AG (CH) 2012-01-11 EP disclosed
WO-2010009402-A9 NILOTINIB INTERMEDIATES AND PREPARATION THEREOF TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2010-06-17 WO disclosed
WO-2010060074-A1 PREPARATION OF NILOTINIB AND INTERMEDIATES THEREOF TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2010-05-27 WO disclosed
WO-2010009402-A2 NILOTINIB INTERMEDIATES AND PREPARATION THEREOF TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2010-01-21 WO disclosed
WO-2007067444-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-06-14 WO disclosed