SCHEMBL10056562

SCHEMBL10056562

N#Cc1ccc(CNC(=O)[C@H](CCCCN)NC(=O)[C@@H](CCCCN)NS(=O)(=O)Cc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
F2 P00734 4/20 0.45
F10 P00742 4/20 0.45
PLG P00747 1/20 0.45
KLKB1 P03952 1/20 0.45
PROC P04070 1/20 0.45
TLR2 O60603 1/20 0.43
PSMB1 P20618 1/20 0.43
PSMB8 P28062 1/20 0.43
PSMB9 P28065 1/20 0.43
PSMB5 P28074 1/20 0.43
PSMB10 P40306 1/20 0.43
PSMB2 P49721 1/20 0.43
NPY1R P25929 7/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15308907 0.87 F2 (0.51) F2F10PLGKLKB1PROC
SCHEMBL321996 0.86 CTSB (0.46) ITGB3ITGA2BF2F10PLG
SCHEMBL10056582 0.84 KLKB1 (0.55) KLKB1
SCHEMBL8347771 0.82 TMPRSS11D (0.58) CA1CA2F2F10PLG
SCHEMBL15308902 0.79 F2 (0.49) F2F10PLGKLKB1PROC
SCHEMBL16821242 0.77 ITGB3 (0.56) CA1CA2ITGB3ITGA2BF2
SCHEMBL16288707 0.76 TLR2 (0.58) CA1CA2TLR2NPY1RNPY5R
SCHEMBL30309011 0.76 ITGB3 (0.65) CA1CA2ITGB3ITGA2BTLR2
SCHEMBL8289977 0.75 F2 (0.61) F2F10PLGKLKB1PROC
SCHEMBL5969435 0.74 ANPEP (0.46) CA1TMPRSS11D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004678-A2 SERINE PROTEASE INHIBITORS THE MEDICINES COMPANY (LEIPZIG) GMBH (DE) 2012-01-12 WO disclosed