SCHEMBL1005841

SCHEMBL1005841

O=[N+]([O-])c1cc([N+](=O)[O-])cc(C(F)(F)F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.55
ALDH1A1 P00352 3/20 0.55
CYP3A4 P08684 3/20 0.55
TDP1 Q9NUW8 2/20 0.55
HPGD P15428 1/20 0.55
ALOX15 P16050 1/20 0.55
HIF1A Q16665 1/20 0.55
TXNRD1 Q16881 1/20 0.55
TXNRD3 Q86VQ6 1/20 0.55
TXNRD2 Q9NNW7 1/20 0.55
CYP19A1 P11511 1/20 0.54
LMNA P02545 1/20 0.46
KIF11 P52732 2/20 0.46
PTPN5 P54829 1/20 0.46
VCAM1 P19320 1/20 0.45
P2RX1 P51575 3/20 0.44
P2RX4 Q99571 1/20 0.44
P2RX7 Q99572 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28212666 0.98 TSHR (0.53) TSHRALDH1A1CYP3A4TDP1HPGD
Hydrazine SCHEMBL28307217 0.96 TSHR (0.52) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL1996062 0.95 ALDH1A1 (0.55) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL29658338 0.87 TSHR (0.48) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL1505899 0.87 TSHR (0.48) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL30600332 0.87 CYP19A1 (0.64) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL2976324 0.86 ALDH1A1 (0.47) TSHRALDH1A1CYP3A4TDP1HPGD
Fluoride SCHEMBL7040657 0.86 ALDH1A1 (0.47) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL788056 0.86 ALDH1A1 (0.47) TSHRALDH1A1CYP3A4TDP1HPGD
SCHEMBL8999953 0.86 ALDH1A1 (0.47) TSHRALDH1A1CYP3A4TDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 182 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928079-A Trefanocide haptens and its preparation method and application 广东第二师范学院 2017-07-07 CN claimed
US-20130177485-A1 DIAGNOSTIC DEVICE FOR IDENTIFYING RUPTURE OF MEMBRANE DURING PREGNANCY MOMTEC LIFE LTD OF YAZMOT HAEMEK (IL) 2013-07-11 US claimed
US-20110065139-A1 DIAGNOSTIC DEVICE FOR IDENTIFYING RUPTURE OF MEMBRANE DURING PREGNANCY MULLERAD JACOB 2011-03-17 US claimed
EP-2198299-A2 A DIAGNOSTIC DEVICE FOR IDENTIFYING RUPTURE OF MEMBRANE DURING PREGNANCY Mullerad, Jacob (IL) 2010-06-23 EP claimed
WO-2009050711-A2 A DIAGNOSTIC DEVICE FOR IDENTIFYING RUPTURE OF MEMBRANE DURING PREGNANCY MULLERAD JACOB (IL) 2009-04-23 WO claimed
WO-2008038042-A1 CHEMICAL PROCESS FOR DISPLACING NITRO GROUPS PHOENIX CHEMICALS LIMITED (GB) 2008-04-03 WO claimed
EP-0413192-A1 Method of making 1,1'-oxybis(3-nitro-5-Trifluoromethyl)benzene OCCIDENTAL CHEMICAL CORPORATION (US) 1991-02-20 EP claimed
US-4990670-A Method of making 1,1'-oxybis (3-nitro-5-trifluoromethyl)-benzene OCCIDENTAL CHEMICAL CORPORATION (US) 1991-02-05 US claimed
EP-0003430-B1 NOVEL 2,6-DINITROBENZENAMINES, THEIR PREPARATION, COMPOSITION CONTAINING THEM AND THEIR USE AS FUNGICIDES ELI LILLY AND COMPANY (US) 1982-01-06 EP claimed
JP-4312544-A None JP disclosed
JP-5286907-A None JP disclosed
JP-6100507-A None JP disclosed
JP-6157428-A None JP disclosed
JP-5085996-A None JP disclosed
EP-0413192-A1 Method of making 1,1'-oxybis(3-nitro-5-Trifluoromethyl)benzene OCCIDENTAL CHEMICAL CORPORATION (US) 1991-02-20 EP disclosed
US-4990670-A Method of making 1,1'-oxybis (3-nitro-5-trifluoromethyl)-benzene OCCIDENTAL CHEMICAL CORPORATION (US) 1991-02-05 US disclosed
US-4876329-A LOW DIELECTRIC CONSTANT, COLORLESS, HEAT STABILITY, HIGH GLASS TRANSITION TEMPERATURE; ELECTRONICS USE AMOCO CORPORATION (US) 1989-10-24 US disclosed
EP-0150587-B1 PREPARATION OF CHLOROBENZOTRIFLUORIDE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-02-03 EP disclosed
EP-0150587-A2 Preparation of chlorobenzotrifluoride compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-08-07 EP disclosed
US-3726930-A PREPARATION OF 3,5-DINITROBENZOTRIFLUORIDE COMPOUNDS UNITED STATES BORAX CHEM 1973-04-10 US disclosed