SCHEMBL10060682

SCHEMBL10060682

Brc1ccc2c(cnn2C2CCNCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM1A O60341 1/20 0.41
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
BRD4 O60885 3/20 0.39
GPR119 Q8TDV5 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
PIM1 P11309 1/20 0.36
PIK3CD O00329 1/20 0.35
SCD O00767 1/20 0.35
TNKS O95271 2/20 0.35
CCR3 P51677 1/20 0.34
PRMT5 O14744 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30450183 1.00 MEN1 (0.43) MEN1ALDH1A1MAPTPKMALOX15
Hydrochloric Acid SCHEMBL30508276 0.98 MEN1 (0.42) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL30508337 0.93 PRMT5 (0.40) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL30508240 0.93 PRMT5 (0.40) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL13468 0.91 HDAC8 (0.39) GPR119HDAC8PIK3CDSCDTNKS
SCHEMBL19703386 0.90 MEN1 (0.42) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL31757809 0.90 MEN1 (0.42) MEN1ALDH1A1MAPTPKMALOX15
Trifluoroacetic Acid SCHEMBL26683826 0.88 HDAC8 (0.41) GPR119HDAC8
SCHEMBL25045382 0.88 HTR7 (0.39) GPR119HDAC8PIK3CDSCDTNKS
SCHEMBL17678127 0.88 PDE9A (0.38) GPR119HDAC8PIK3CDSCDTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146035-A1 FUSED BICYCLIC COMPOUNDS AND THEIR USE AS MER AND AXL INHIBITORS DONG-A ST CO., LTD. (KR) 2026-05-28 US disclosed
EP-4605395-A2 FUSED BICYCLIC COMPOUNDS AND THEIR USE AS MER AND AXL INHIBITORS Dong-A ST Co., Ltd. (KR) 2025-08-27 EP disclosed
WO-2024084448-A2 FUSED BICYCLIC COMPOUNDS AND THEIR USE AS MER AND AXL INHIBITORS DONG-A ST CO., LTD. (KR) 2024-04-25 WO disclosed
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
US-20230374007-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-11-23 US disclosed
US-20230374007-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-11-23 US disclosed
US-20230374007-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-11-23 US disclosed
WO-2023198114-A1 ALK2 KINASE INHIBITOR 杭州邦顺制药有限公司 2023-10-19 WO disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed
EP-2837623-A1 NOVEL 1-SUBSTITUTED INDAZOLE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2015-02-18 EP disclosed
WO-2012086735-A1 CONDENSED HETEROCYCLIC COMPOUND 大正製薬株式会社 (JP) 2012-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260146035-A1 FUSED BICYCLIC COMPOUNDS AND THEIR USE AS MER AND AXL INHIBITORS AXL, ERBB2, ERBB3 MEN1 2419/4885ALDH1A1 2378/4885MAPT 3785/4885
US-20230374007-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER RARA, RARG, RARB MEN1 153/4885ALDH1A1 72/4885MAPT 3773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.