SCHEMBL10065013

SCHEMBL10065013

CCOC(=O)c1c(-c2ccccc2C=O)c2ccccc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 4/20 0.43
NOD1 Q9Y239 4/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 2/20 0.41
AR P10275 1/20 0.41
NTRK1 P04629 1/20 0.40
RECQL P46063 1/20 0.40
AGTR1 P30556 3/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ELANE P08246 1/20 0.39
UBE2N P61088 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10065051 0.86 PSEN1 (0.40) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL11901256 0.79 NOD2 (0.56) NOD2NOD1MEN1KMT2AAR
SCHEMBL12229940 0.78 NOD2 (0.49) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL12392496 0.76 NOD2 (0.48) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL13765387 0.74 NOD2 (0.46) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL8874979 0.72 NOD2 (0.49) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL2732415 0.72 MEN1 (0.45) MEN1KMT2APSEN1PSEN2APH1B
SCHEMBL7467719 0.71 NOD2 (0.57) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL13765375 0.71 MEN1 (0.45) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL2005697 0.69 NOD2 (0.53) NOD2NOD1ALDH1A1ALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed