SCHEMBL2732415

SCHEMBL2732415

O=Cc1ccccc1-c1c(C(=O)O)n(S(=O)(=O)c2ccccc2)c2ccc(OCc3ccccc3)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
EDNRB P24530 4/20 0.44
EDNRA P25101 4/20 0.44
HTR6 P50406 2/20 0.43
LTB4R Q15722 1/20 0.43
ACLY P53396 1/20 0.42
BCL2 P10415 1/20 0.41
BID P55957 1/20 0.41
MCL1 Q07820 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
SRD5A2 P31213 1/20 0.39
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP12 P39900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2732313 0.84 HTR6 (0.39) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL2732312 0.84 HTR6 (0.39) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL2733167 0.83 HTR6 (0.40) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL2732065 0.81 HTR6 (0.42) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL2733056 0.81 HTR6 (0.42) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL2731882 0.80 HTR6 (0.48) MEN1NPC1RAB9AKMT2AEDNRB
SCHEMBL10065051 0.80 PSEN1 (0.40) MEN1KMT2AHTR6PSEN1PSEN2
SCHEMBL2886894 0.74 HTR6 (0.63) MEN1NPC1RAB9AKMT2AHTR6
SCHEMBL8857175 0.74 EDNRA (0.62) EDNRBEDNRA
SCHEMBL10065013 0.72 NOD2 (0.43) MEN1KMT2AHTR6PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed