SCHEMBL10066965

SCHEMBL10066965

Cc1cncc(-c2ncc(C(=O)NCc3cccc(C(N)=O)c3)s2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.53
ROCK2 O75116 9/20 0.50
PPARA Q07869 1/20 0.44
ENPP2 Q13822 1/20 0.43
ROCK1 Q13464 2/20 0.43
BMPR2 Q13873 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
GSK3B P49841 2/20 0.40
KLKB1 P03952 1/20 0.40
WDR5 P61964 1/20 0.40
MMP13 P45452 1/20 0.39
P2RX7 Q99572 1/20 0.39
DYRK3 O43781 1/20 0.39
PRKCG P05129 1/20 0.39
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
MAPK1 P28482 1/20 0.39
CLK2 P49760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10066502 0.84 ROCK2 (0.61) F10ROCK2PPARAENPP2ROCK1
SCHEMBL10066964 0.82 F10 (0.52) F10ROCK2ENPP2ROCK1BMPR2
SCHEMBL10022593 0.77 ROCK2 (0.80) ROCK2
SCHEMBL4897260 0.72 ESRRG (0.54) ROCK2PPARAROCK1
SCHEMBL12788248 0.72 PPARA (0.69) PPARAMMP13
SCHEMBL13068789 0.72 MMP13 (0.59) F10ROCK2ROCK1MMP13
SCHEMBL13947481 0.71 MMP13 (0.60) F10ROCK2ROCK1KLKB1MMP13
SCHEMBL12697566 0.69 PPARA (0.47) PPARAMMP13P2RX7
SCHEMBL4896887 0.69 HDAC3 (0.56) ROCK2PPARAROCK1GSK3BDYRK3
SCHEMBL10022672 0.69 HCAR2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006203-A1 N-CYCLYL-3 - (CYCLYLCARBONYLAMINOMETHYL) BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed