SCHEMBL10066964

SCHEMBL10066964

Cc1ccncc1-c1ncc(C(=O)NCc2cccc(C(N)=O)c2)s1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.52
ROCK2 O75116 11/20 0.49
BMPR2 Q13873 2/20 0.46
ENPP2 Q13822 1/20 0.43
ROCK1 Q13464 3/20 0.42
GSK3B P49841 1/20 0.41
NPC1 O15118 1/20 0.41
WDR5 P61964 1/20 0.41
F2 P00734 1/20 0.40
GRK2 P25098 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10066965 0.82 F10 (0.53) F10ROCK2BMPR2ENPP2ROCK1
SCHEMBL10066502 0.82 ROCK2 (0.61) F10ROCK2BMPR2ENPP2ROCK1
SCHEMBL10022702 0.77 ROCK2 (0.68) ROCK2
SCHEMBL10022599 0.77 ROCK2 (0.76) ROCK2ROCK1
SCHEMBL10022673 0.70 HCAR2 (0.49) NPC1
SCHEMBL27817481 0.69 CDC7 (0.49) NPC1
SCHEMBL27605419 0.69 CDC7 (0.45) NPC1
SCHEMBL13068789 0.69 MMP13 (0.59) F10ROCK2ROCK1
SCHEMBL28595774 0.68 CDC7 (0.69) GSK3B
SCHEMBL3647370 0.68 ALDH1A1 (0.64) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006203-A1 N-CYCLYL-3 - (CYCLYLCARBONYLAMINOMETHYL) BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed