SCHEMBL10067301

SCHEMBL10067301

CN(C)S(=O)(=O)c1ccc2[nH]c(Cl)c(-c3nc4c5cccnc5c5ncccc5c4[nH]3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.38
MEN1 O00255 1/20 0.37
CLK1 P49759 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
PLA2G1B P04054 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
POLB P06746 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
HTR6 P50406 1/20 0.35
PTPN11 Q06124 1/20 0.35
JAK2 O60674 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067318 0.87 RXFP1 (0.34) PTGESMEN1CLK1KMT2AKDM4E
SCHEMBL10067259 0.81 PTGES (0.44) PTGESKDM4EALDH1A1HPGDJAK2
SCHEMBL10082885 0.80 RHEB (0.37) PTGESALDH1A1JAK2CDK4CCND1
SCHEMBL10067303 0.80 EGFR (0.44) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL10067282 0.73 MAP3K14 (0.50) PTGESMEN1KMT2AKDM4EALDH1A1
SCHEMBL10067391 0.70 KDM4E (0.45) PTGESMEN1KMT2AKDM4EALDH1A1
SCHEMBL10082076 0.70 ALDH1A1 (0.35) PTGESMEN1KMT2AKDM4EALDH1A1
SCHEMBL21180305 0.69 SCD (0.47) PTGESALDH1A1SMN1; SMN2PTGS2
SCHEMBL10067256 0.69 MEN1 (0.56) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL10067288 0.69 GABRA1 (0.47) MEN1KMT2AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8148392-B2 2-indolyl imidazo [4,5-d] phenanthroline derivatives and their use in the treatment of cancer LORUS THERAPEUTICS INC. (CA) 2012-04-03 US disclosed
US-20100168417-A1 2-Indolyl Imidazo [4,5-d] Phenanthroline Derivatives and Their Use in the Treatment for Cancer APTOSE BIOSCIENCES INC. (CA) 2010-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168417-A1 2-Indolyl Imidazo [4,5-d] Phenanthroline Derivatives and Their Use in the Treatment for Cancer FLI1, IKZF3, IKZF2 PTGES 1934/4885MEN1 2366/4885CLK1 2700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.