SCHEMBL10067397

SCHEMBL10067397

O=C(NCC1CCCC1)c1nc(C2CN=CN2c2cccc(F)c2F)c[nH]1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.40
ADORA1 P30542 1/20 0.40
AR P10275 1/20 0.36
CNR1 P21554 3/20 0.35
GSK3B P49841 3/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CNR2 P34972 3/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KCNH2 Q12809 2/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
JAK3 P52333 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600764 0.75 ADORA2A (0.40) ADORA2AADORA1ARCNR1GSK3B
SCHEMBL14600762 0.75 ADORA2A (0.40) ADORA2AADORA1ARCNR1GSK3B
SCHEMBL14600758 0.69 GSK3B (0.41) ADORA2AADORA1ARCNR1GSK3B
SCHEMBL14600765 0.69 ADORA2A (0.41) ADORA2AADORA1ARCNR1CCNA2
SCHEMBL14286135 0.65 ROCK2 (0.41) ADORA2AADORA1GSK3BCCNA2CDK2
SCHEMBL14286139 0.65 ROCK2 (0.40) ADORA2AADORA1GSK3BCCNA2CDK2
SCHEMBL10067974 0.64 CHRM1 (0.40) ADORA2AADORA1ARCNR1CCNA2
SCHEMBL14600763 0.64 GSK3B (0.44) GSK3BKCNH2KMT2AMEN1
SCHEMBL10067975 0.64 ALDH1A1 (0.46) GSK3BKCNH2KMT2AMEN1
SCHEMBL10067976 0.64 GSK3B (0.44) GSK3BKCNH2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697352-B1 4-AZOLE SUBSTITUTED IMIDAZOLE COMPOSITIONS USEFUL AS INHIBITORS OR C-MET RECEPTOR TYROSINE KINASE VERTEX PHARMA (US) 2012-06-27 EP disclosed