SCHEMBL10067971

SCHEMBL10067971

C=C(NCCCn1ccnc1)c1nc(-c2oncc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
TSHR P16473 2/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
ADORA2A P29274 1/20 0.37
QPCT Q16769 6/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NAMPT P43490 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600776 0.91 ALDH1A1 (0.46) ALDH1A1TSHRHSP90AA1HSP90AB1ADORA2A
SCHEMBL14600751 0.86 GAA (0.46) ALDH1A1TSHRHSP90AA1HSP90AB1ADORA2A
SCHEMBL14286125 0.76 ADORA2A (0.53) ALDH1A1TSHRHSP90AA1HSP90AB1ADORA2A
SCHEMBL14600757 0.75 ALDH1A1 (0.44) ALDH1A1TSHRHSP90AA1HSP90AB1ADORA2A
SCHEMBL14600775 0.67 BCAT1 (0.39) POLBSMN1; SMN2
SCHEMBL5565224 0.67 BCAT1 (0.37)
SCHEMBL14600777 0.66 GSK3B (0.53) ALDH1A1POLBMEN1KMT2AGAA
SCHEMBL14286129 0.64 ADORA2A (0.53) ALDH1A1ADORA2APOLBMEN1KMT2A
SCHEMBL5047841 0.63 ADORA2A (0.53) ALDH1A1TSHRADORA2APOLBMEN1
SCHEMBL4831524 0.63 BCAT1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697352-B1 4-AZOLE SUBSTITUTED IMIDAZOLE COMPOSITIONS USEFUL AS INHIBITORS OR C-MET RECEPTOR TYROSINE KINASE VERTEX PHARMA (US) 2012-06-27 EP disclosed