SCHEMBL14600751

SCHEMBL14600751

O=C(NCCCn1ccnc1)c1nc(-c2cnoc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
ADORA2A P29274 1/20 0.45
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NAMPT P43490 2/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 2/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 2/20 0.43
HTT P42858 1/20 0.43
HIF1A Q16665 1/20 0.43
TSHR P16473 2/20 0.43
HSP90AA1 P07900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600776 0.95 ALDH1A1 (0.46) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL10067971 0.86 ALDH1A1 (0.38) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL14286125 0.85 ADORA2A (0.53) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL14600757 0.84 ALDH1A1 (0.44) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL14600753 0.74 GSK3B (0.53) GAAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL14600755 0.72 BCAT1 (0.41) POLBRAB9ANPC1
SCHEMBL14286129 0.71 ADORA2A (0.53) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL5047841 0.70 ADORA2A (0.53) GAAADORA2AALDH1A1CYP1A2CYP3A4
SCHEMBL1179031 0.69 GLA (0.75) GAAALDH1A1CYP3A4CYP2C19NAMPT
SCHEMBL14600777 0.68 GSK3B (0.53) GAAALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed