SCHEMBL10068053

SCHEMBL10068053

CS(=O)(=O)c1ccc(-c2cc(F)c(OCC3C4CN(C#N)C[C@H]34)c(F)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.39
PTGS2 P35354 10/20 0.38
KIF11 P52732 1/20 0.38
PTGS1 P23219 1/20 0.37
LRRK2 Q5S007 2/20 0.36
UCHL1 P09936 1/20 0.36
CTSK P43235 1/20 0.36
CTSC P53634 1/20 0.36
BRD4 O60885 1/20 0.36
USP30 Q70CQ3 1/20 0.35
NAAA Q02083 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903884 0.81 KIF11 (0.41) PTGS2KIF11PTGS1BRD4
SCHEMBL903936 0.79 GPR119 (0.48)
SCHEMBL10067699 0.79 NR1H2 (0.40) PTGS2KIF11PTGS1
SCHEMBL904082 0.78 GPR119 (0.47) PTGS2
SCHEMBL903891 0.78 GPR119 (0.47) PTGS2
SCHEMBL10067702 0.77 GPR119 (0.45) PTGS2
SCHEMBL10068069 0.77 GPR119 (0.45) PTGS2
SCHEMBL903897 0.76 GPR119 (0.40) PTGS2KIF11PTGS1
SCHEMBL10067575 0.76 GPR119 (0.47) PTGS2PTGS1LRRK2
SCHEMBL904103 0.75 NR1H2 (0.41) PTGS2NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed