Acridine

Acridine

SCHEMBL1006962

N=C=S.c1ccc2nc3ccccc3cc2c1.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.71
HPGD P15428 3/20 0.71
MAPT P10636 3/20 0.71
GLA P06280 2/20 0.71
ACHE P22303 1/20 0.71
HTR3A P46098 1/20 0.52
NQO2 P16083 2/20 0.48
KDM4E B2RXH2 3/20 0.45
GAA P10253 3/20 0.45
KMT2A Q03164 3/20 0.45
NPC1 O15118 3/20 0.45
POLB P06746 2/20 0.45
RAB9A P51151 2/20 0.45
LMNA P02545 1/20 0.45
PTBP1 P26599 1/20 0.45
RCE1 Q9Y256 1/20 0.45
TDP1 Q9NUW8 1/20 0.42
STAT3 P40763 1/20 0.42
PDE10A Q9Y233 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL37657 1.00 ALDH1A1 (0.71) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL28002752 0.86 ALDH1A1 (0.71) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL10533085 0.86 ALDH1A1 (0.71) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL1772714 0.84 ALDH1A1 (1.00) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL4972293 0.84 ALDH1A1 (1.00) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL29352289 0.84 ALDH1A1 (1.00) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL8339 0.84 ALDH1A1 (1.00) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL3045498 0.84 ALDH1A1 (1.00) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL1551975 0.82 ALDH1A1 (0.94) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL2394207 0.82 ALDH1A1 (0.94) ALDH1A1HPGDMAPTGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021263188-A9 LIVE CELL ENGAGEMENT ASSAY ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-06-09 WO disclosed
WO-2021263188-A1 LIVE CELL ENGAGEMENT ASSAY ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2021-12-30 WO disclosed
EP-2268608-A2 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES Biosearch Technologies, Inc. (US) 2011-01-05 EP disclosed
WO-2009152102-A2 PRO-FLUORESCENT PROBES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-12-17 WO disclosed
EP-2114905-A1 MULTI-COLOR TIME RESOLVED FLUOROPHORES BASED ON MACROCYCLIC LANTHANIDE COMPLEXES Lumiphore, Inc. (US) 2009-11-11 EP disclosed
WO-2009124150-A2 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES BIOSEARCH TECHNOLOGIES, INC. (US) 2009-10-08 WO disclosed
EP-1896613-A4 NON-IN SITU HYBRIDIZATION METHOD FOR DETECTING CHROMOSOMAL ABNORMALITIES QUEST DIAGNOSTICS INVEST INC (US) 2009-09-02 EP disclosed
EP-2082055-A2 NUCLEIC ACID SIZE DETECTION METHOD Quest Diagnostics Investments Incorporated (US) 2009-07-29 EP disclosed
EP-1766061-A4 SINGLE LABEL COMPARATIVE HYBRIDIZATION QUEST DIAGNOSTICS INVEST INC (US) 2009-05-27 EP disclosed
EP-2051968-A2 LUMINESCENT MACROCYCLIC LANTHANIDE COMPLEXES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-04-29 EP disclosed
EP-1305445-A4 DARK QUENCHERS FOR DONOR-ACCEPTOR ENERGY TRANSFER BIOSEARCH TECHNOLOGIES INC (US) 2003-08-13 EP disclosed
EP-1305445-A1 DARK QUENCHERS FOR DONOR-ACCEPTOR ENERGY TRANSFER Biosearch Technologies, Inc. (US) 2003-05-02 EP disclosed
WO-2003000933-A1 DUAL RESONANCE ENERGY TRANSFER NUCLEIC ACID PROBES GEORGIA TECH RESEARCH CORPORATION (US) 2003-01-03 WO disclosed
WO-2002057479-A2 PRIMERS AND METHODS FOR THE DETECTION AND DISCRIMINATION OF NUCLEIC ACIDS INVITROGEN CORPORATION (US) 2002-07-25 WO disclosed
WO-2000079009-A9 IMPROVED PRIMERS AND METHODS FOR THE DETECTION AND DISCRIMINATION OF NUCLEIC ACIDS INVITROGEN CORP (US) 2002-06-13 WO disclosed
WO-2002044399-A2 IN VITRO TRANSCRIPTION METHOD FOR RNA AMPLIFICATION ROSETTA INPHARMATICS, INC. (US) 2002-06-06 WO disclosed
WO-2002026867-A2 DENDRIMERIC SUPPORT OR CARRIER MACROMOLECULE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-04-04 WO disclosed
EP-1190097-A2 IMPROVED PRIMERS AND METHODS FOR THE DETECTION AND DISCRIMINATION OF NUCLEIC ACIDS INVITROGEN CORPORATION (US) 2002-03-27 EP disclosed
WO-2001086001-A1 DARK QUENCHERS FOR DONOR-ACCEPTOR ENERGY TRANSFER BIOSEARCH TECHNOLOGIES, INC. (US) 2001-11-15 WO disclosed
WO-2000079009-A2 IMPROVED PRIMERS AND METHODS FOR THE DETECTION AND DISCRIMINATION OF NUCLEIC ACIDS INVITROGEN CORPORATION (US) 2000-12-28 WO disclosed