SCHEMBL10069653

SCHEMBL10069653

Bc1cnc(N)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.39
MAP3K12 Q12852 11/20 0.38
PIK3CD O00329 1/20 0.38
TNF P01375 1/20 0.36
PIK3CA P42336 5/20 0.35
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21031807 0.78 GLA (0.45) MTORMAP3K12PIK3CDTNFPIK3CA
SCHEMBL29601287 0.78 GLA (0.45) MTORMAP3K12PIK3CDTNFPIK3CA
SCHEMBL18072106 0.77 MTOR (0.40) MTORMAP3K12PIK3CDTNFPIK3CA
SCHEMBL3643010 0.77 ALDH1A1 (0.43) MTORMAP3K12TNFPIK3CAPOLB
SCHEMBL503280 0.75 IDO1 (0.43) MTORMAP3K12PIK3CDTNFPIK3CA
SCHEMBL17619923 0.75 HPGD (0.32) PIK3CD
SCHEMBL182671 0.75 HTT (0.54) MTORMAP3K12TNFPIK3CAPOLB
SCHEMBL11890838 0.75 NOS3 (0.54) MTORMAP3K12PIK3CDPIK3CA
SCHEMBL13186700 0.75 PIK3CD (0.34) PIK3CD
SCHEMBL1583813 0.75 IDO1 (0.43) MTORMAP3K12PIK3CDTNFPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925757-B1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2017-10-04 EP disclosed
WO-2012034526-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2012-03-22 WO disclosed
WO-2010091409-A1 CERTAIN NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GLAXOSMITHKLINE LLC (US) 2010-08-12 WO disclosed