SCHEMBL10072039

SCHEMBL10072039

O=C(Nc1ccccc1N1CCCCC1)C1CC12CCN(Cc1ccccc1)CC2

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.63
KCNQ2 O43526 5/20 0.52
KMT2A Q03164 4/20 0.52
GAA P10253 2/20 0.52
PKM P14618 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52
CSF1R P07333 3/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
LMNA P02545 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
PLA2G1B P04054 1/20 0.45
ATM Q13315 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709233 0.82 ALDH1A1 (0.51) KMT2AGAAALDH1A1TSHRNPSR1
SCHEMBL1709232 0.78 SCN9A (1.00) SCN9AKCNQ2KMT2AGAAPKM
SCHEMBL7540788 0.71 ALDH1A1 (0.55) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL13167010 0.69 KCNQ2 (1.00) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL4318899 0.68 KCNQ2 (0.68) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL2796459 0.68 HRH3 (1.00) KMT2AHRH3ALDH1A1MEN1KDM4E
SCHEMBL29559749 0.68 KCNQ2 (0.68) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL29957640 0.68 KMT2A (0.72) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL22897679 0.68 KCNQ2 (0.68) KCNQ2KMT2AGAAPKMALDH1A1
SCHEMBL18838361 0.67 HRH3 (0.51) KMT2APKMHRH3MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed