SCHEMBL10072404

SCHEMBL10072404

CCN1CCN(CCCCc2c[nH]c3ccc(F)cc23)CC1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.81
MPO P05164 5/20 0.78
SLC6A4 P31645 3/20 0.67
HTR7 P34969 2/20 0.62
KCNH2 Q12809 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763035 0.87 HTR1A (0.76) HTR1AMPOSLC6A4HTR7KCNH2
SCHEMBL739944 0.86 HTR1A (0.79) HTR1AMPOSLC6A4
SCHEMBL4261226 0.85 HTR1A (0.76) HTR1AMPOSLC6A4
SCHEMBL6347575 0.84 HTR1A (0.74) HTR1AMPOSLC6A4
SCHEMBL16441164 0.82 HTR1A (1.00) HTR1AMPO
SCHEMBL9047205 0.82 HTR1A (0.85) HTR1AMPOSLC6A4HTR7KCNH2
SCHEMBL27836200 0.82 MPO (1.00) HTR1AMPOSLC6A4HTR7
SCHEMBL9368593 0.82 HTR1A (0.92) HTR1AMPOSLC6A4HTR7KCNH2
SCHEMBL8557097 0.81 HTR1A (0.70) HTR1AMPOSLC6A4HTR7KCNH2
SCHEMBL16432976 0.81 HTR1A (1.00) HTR1ASLC6A4HTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138174-B2 Such as N-{1-[7-(2-amino-ethoxyimino)-7-[4-(trifluoromethyl)phenyl]heptylamino]-1-[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-methylidene)-4-chloro-benzenesulfonamide; pain. psychosis, anxiety, depression, attention deficits, cognitive disorders, obesity; neurodegenerative disorders SOLVAY PHARMACEUTICALS B.V. (NL) 2012-03-20 US disclosed