SCHEMBL10074293

SCHEMBL10074293

CC(C)(CNC(=O)C[C@H](N)Cc1cc(F)ccc1F)CNC(=O)[C@@H](O)[C@H](N)CO

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.43
DPP8 Q6V1X1 12/20 0.43
DPP7 Q9UHL4 6/20 0.42
REN P00797 1/20 0.39
DPP9 Q86TI2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10077381 1.00 DPP4 (0.43) DPP4DPP8DPP7RENDPP9
SCHEMBL10074292 1.00 DPP4 (0.43) DPP4DPP8DPP7RENDPP9
SCHEMBL10074134 1.00 DPP4 (0.43) DPP4DPP8DPP7RENDPP9
SCHEMBL10074283 0.90 REN (0.37) DPP4DPP8DPP7RENDPP9
SCHEMBL6874726 0.89 REN (0.41) DPP4DPP8DPP7RENDPP9
SCHEMBL6873681 0.89 LAP3 (0.44) DPP4DPP8DPP7RENDPP9
SCHEMBL13194653 0.89 REN (0.41) DPP4DPP8DPP7RENDPP9
SCHEMBL13194656 0.88 DPP4 (0.41) DPP4DPP8DPP7RENDPP9
SCHEMBL10078068 0.86 METAP2 (0.45) DPP4DPP8DPP7RENDPP9
SCHEMBL6872762 0.86 LAP3 (0.40) DPP4DPP8DPP7RENDPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418196-A1 Dual alanyl-aminopeptidase and dipeptidyl-peptidase IV inhibitors IMTM GmbH (DE) 2012-02-15 EP disclosed