SCHEMBL10074706

SCHEMBL10074706

C[C@H]1CCc2cc3nc(CO)[nH]c(=O)c3cc21

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.37
PARP14 Q460N5 6/20 0.35
KDM4E B2RXH2 3/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HCAR2 Q8TDS4 1/20 0.34
RECQL P46063 1/20 0.34
ALOX12 P18054 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067671 0.85 ALDH1A1 (0.42) PARP14KDM4EGAAMAPTMEN1
SCHEMBL13842610 0.81 QTRT1 (0.41)
SCHEMBL15180107 0.78 PARP1 (0.39) PARP1PARP14KDM4EMAPTMEN1
SCHEMBL10209809 0.78 TNKS2 (0.45) PARP1PARP14KDM4EGAAMAPT
SCHEMBL15180115 0.78 TNKS2 (0.45) PARP1PARP14KDM4EGAAMAPT
SCHEMBL989078 0.77 GRIN2D (0.40) PARP1PARP14KDM4EGAAMAPT
SCHEMBL6585979 0.75 KDM4E (0.41) PARP1PARP14KDM4ERECQL
SCHEMBL3674777 0.74 KDM4E (0.43) PARP1PARP14KDM4EMAPTMEN1
SCHEMBL3674775 0.74 KDM4E (0.43) PARP1PARP14KDM4EMAPTMEN1
SCHEMBL431949 0.74 MAPT (0.37) PARP1PARP14KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087888-A2 EFFICIENT PEPTIDE COUPLINGS AND THEIR USE IN THE SYNTHESIS AND ISOLATION OF A CYCLOPENTA (G) QUINAZOLINE TRISODIUM SALT ONYX PHARMACEUTICALS, INC. (US) 2012-06-28 WO disclosed