SCHEMBL10074721

SCHEMBL10074721

O=C(NC(Cc1ccc(-c2cccnc2)cc1)C(O)C(=O)O)OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.50
CYP3A4 P08684 2/20 0.49
PPARA Q07869 1/20 0.48
TRPM8 Q7Z2W7 1/20 0.47
ITGA4 P13612 1/20 0.45
ITGB7 P26010 1/20 0.45
MMP12 P39900 1/20 0.45
CTRB1 P17538 2/20 0.45
TACR1 P25103 3/20 0.44
ECE1 P42892 1/20 0.44
MAPK1 P28482 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGAV P06756 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435563 0.90 PPARA (0.56) PPARATRPM8CTRB1TACR1ITGB3
SCHEMBL10054485 0.90 CYP3A4 (0.51) NAAACYP3A4TRPM8MMP12MAPK1
SCHEMBL6350990 0.84 TRPM8 (0.61) TRPM8CTRB1TACR1ITGB3
SCHEMBL7414480 0.84 TRPM8 (0.61) TRPM8CTRB1TACR1ITGB3
SCHEMBL7418088 0.84 TRPM8 (0.61) TRPM8CTRB1TACR1ITGB3
SCHEMBL7430937 0.84 TRPM8 (0.61) TRPM8CTRB1TACR1ITGB3
SCHEMBL7245549 0.84 TRPM8 (0.61) TRPM8CTRB1TACR1ITGB3
SCHEMBL3798084 0.82 CYP3A4 (0.52) NAAACYP3A4MMP12CTRB1TACR1
SCHEMBL3798080 0.82 CYP3A4 (0.52) NAAACYP3A4MMP12CTRB1TACR1
SCHEMBL10054482 0.82 NAAA (0.46) NAAACYP3A4PPARATRPM8ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418196-A1 Dual alanyl-aminopeptidase and dipeptidyl-peptidase IV inhibitors IMTM GmbH (DE) 2012-02-15 EP disclosed