SCHEMBL10078712

SCHEMBL10078712

Cc1cc2c(o1)CNCCC2Oc1ccc(C#N)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.40
IMPDH1 P20839 1/20 0.40
CYP3A4 P08684 1/20 0.36
ESRRA P11474 1/20 0.36
PNMT P11086 1/20 0.33
AR P10275 5/20 0.31
HTR6 P50406 2/20 0.31
HTR2A P28223 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2835872 0.99 IMPDH2 (0.39) IMPDH2IMPDH1CYP3A4ESRRAPNMT
SCHEMBL10078641 0.86 HTR2C (0.33)
SCHEMBL10078500 0.84 PKM (0.31)
Hydrochloric Acid SCHEMBL2841127 0.83 PKM (0.30)
SCHEMBL2844093 0.82 IMPDH2 (0.39) IMPDH2IMPDH1CYP3A4ESRRAPNMT
SCHEMBL2840787 0.82 SLC6A2 (0.38) HTR6
Hydrochloric Acid SCHEMBL3570724 0.81 IMPDH2 (0.39) IMPDH2IMPDH1CYP3A4ESRRAPNMT
Hydrochloric Acid SCHEMBL2837096 0.81 SLC6A2 (0.37) HTR6
Hydrochloric Acid SCHEMBL2868875 0.76 HTR2C (0.34)
SCHEMBL10078928 0.73 SLC6A4 (0.40) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US claimed