SCHEMBL10083012

SCHEMBL10083012

Nc1ccc(C2(C(=O)O)CC2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.47
GABRD O14764 2/20 0.47
GABRA1 P14867 2/20 0.47
GABRB1 P18505 2/20 0.47
GABRG2 P18507 2/20 0.47
GABRB3 P28472 2/20 0.47
GABRA5 P31644 2/20 0.47
GABRA3 P34903 2/20 0.47
GABRA2 P47869 2/20 0.47
GABRB2 P47870 2/20 0.47
GABRA4 P48169 2/20 0.47
GABRE P78334 2/20 0.47
GABRA6 Q16445 2/20 0.47
GABRG1 Q8N1C3 2/20 0.47
GABRG3 Q99928 2/20 0.47
GABRQ Q9UN88 2/20 0.47
AKR1C1 Q04828 2/20 0.43
NNMT P40261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAP4K4 O95819 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL349552 0.79 NAPRT (0.47) AKR1C1SMN1; SMN2MAP4K4AKR1C3AKR1C2
SCHEMBL31247665 0.79 NAPRT (0.47) AKR1C1SMN1; SMN2MAP4K4AKR1C3AKR1C2
SCHEMBL350673 0.75 AKR1C1 (0.55) AKR1C1MAP4K4ALDH1A1AKR1C3AKR1C2
SCHEMBL3258917 0.75 NNMT (0.46) AKR1C1NNMTKDM4EALDH1A1MEN1
SCHEMBL1951679 0.75 MAP4K4 (0.54) AKR1C1MAP4K4AKR1C3AKR1C2MEN1
SCHEMBL14872334 0.75 KMT2A (0.46) AKR1C1MAP4K4AKR1C3AKR1C2MEN1
SCHEMBL348598 0.75 LDHA (0.51) AKR1C1AKR1C3AKR1C2
SCHEMBL14868369 0.75 AKR1C1 (0.40) AKR1C1MAP4K4AKR1C3AKR1C2MEN1
SCHEMBL12138123 0.74 MAP4K4 (0.40) AKR1C1MAP4K4KDM4EALDH1A1GAA
SCHEMBL17298724 0.73 NOS3 (0.40) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed