SCHEMBL1008927

SCHEMBL1008927

N=C(N)NCCC[C@H](N)C(=O)Nc1ccc(C(=O)O)c(C(=O)c2ccccc2)c1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10710806 0.84 KDM4C (0.44)
Hydrochloric Acid SCHEMBL10713210 0.83 KDM4C (0.44)
SCHEMBL8768680 0.81 LTA4H (0.47)
SCHEMBL2033471 0.80 LNPEP (0.44)
SCHEMBL2585866 0.79 EPHX1 (0.47)
SCHEMBL29359776 0.79 EPHX1 (0.47)
SCHEMBL19445842 0.78 POLB (0.52)
Hydrochloric Acid SCHEMBL4087778 0.78 EPHX1 (0.46)
SCHEMBL14250016 0.78 CYP2C9 (0.46)
SCHEMBL9335651 0.76 EPHX2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268654-A2 SELECTIVE HIGH-AFFINITY POLYDENTATE LIGANDS AND METHODS OF MAKING SUCH The Regents of the University of California (US) 2011-01-05 EP disclosed
WO-2009132020-A2 SELECTIVE HIGH-AFFINITY POLYDENTATE LIGANDS AND METHODS OF MAKING SUCH THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-10-29 WO disclosed