SCHEMBL10089928

SCHEMBL10089928

Cc1cc(Cl)cc(C(=O)NC2CCN(C)CC2)c1NC(=O)c1cc(Cn2nnc(C(F)(F)F)n2)nn1-c1ncccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 4/20 0.35
CRHR1 P34998 5/20 0.35
MAPK14 Q16539 2/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
NTRK1 P04629 4/20 0.33
SSTR1 P30872 1/20 0.33
MALT1 Q9UDY8 1/20 0.33
JAK2 O60674 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL685487 0.95 CRHR1 (0.38) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL13085060 0.94 CRHR1 (0.36) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10089868 0.93 NTRK1 (0.36) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10089957 0.92 CRHR1 (0.35) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10089845 0.91 NTRK1 (0.34) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10089471 0.91 DRD4 (0.42)
SCHEMBL10089862 0.91 DGAT2 (0.36) CRHR1NTRK1
SCHEMBL13085405 0.90 CRHR1 (0.37) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL686481 0.90 CRHR1 (0.36) CRHR1MAPK14MAPK13MAPK12MAPK11
SCHEMBL13085179 0.90 CRHR1 (0.38) CRHR1MAPK14MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8791143-B2 Anthranilic diamide derivatives having cyclic side-chains BAYER CROPSCIENCE AG (DE) 2014-07-29 US disclosed
US-20120010249-A1 Anthranilic diamide derivatives having cyclic side-chains BAYER CROPSCIENCE AG (DE) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010249-A1 Anthranilic diamide derivatives having cyclic side-chains DDT, ADCY1, ANTXR2 SSTR4 3131/4885CRHR1 3984/4885MAPK14 2788/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.