SCHEMBL10090899

SCHEMBL10090899

CN(C)CCCn1ccnn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.38
CYP2D6 P10635 5/20 0.36
CYP19A1 P11511 2/20 0.36
ALDH1A1 P00352 4/20 0.35
LMNA P02545 3/20 0.35
MAPT P10636 3/20 0.35
CYP1A2 P05177 3/20 0.35
SLC22A1 O15245 2/20 0.35
PRNP P04156 2/20 0.35
CHRM2 P08172 2/20 0.35
CHRM4 P08173 2/20 0.35
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
DRD2 P14416 2/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
CHRM3 P20309 2/20 0.35
DRD1 P21728 2/20 0.35
DRD4 P21917 2/20 0.35
DRD5 P21918 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10065550 0.88 HTR1A (0.40) HTR1ACYP19A1HTR2AHTR2CKDM1A
SCHEMBL27085532 0.77
SCHEMBL27085525 0.75 CYP19A1 (0.42) CYP19A1DPP4ATP4AATP4B
SCHEMBL628307 0.75 TBXAS1 (0.42) CYP19A1ALDH1A1LMNAMAPTSMPD1
SCHEMBL11361006 0.75 CYP19A1 (0.48) CYP19A1ALDH1A1KMT2ADPP4
SCHEMBL6071635 0.74
SCHEMBL11204798 0.73 TBXAS1 (0.46) CYP19A1LMNAMAPTSMPD1KDM4E
SCHEMBL243704 0.73 TBXAS1 (0.46) CYP19A1LMNAMAPTSMPD1KDM4E
SCHEMBL21925549 0.73 TBXAS1 (0.46) CYP19A1LMNAMAPTSMPD1KDM4E
SCHEMBL3302887 0.73 TBXAS1 (0.46) CYP19A1LMNAMAPTSMPD1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160152814-A1 4- AND 5-SUBSTITUTED 1,2,3-TRIAZOLE, AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS ISP INVESTMENTS INC. (US) 2016-06-02 US disclosed
US-20160152814-A1 4- AND 5-SUBSTITUTED 1,2,3-TRIAZOLE, AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS ISP INVESTMENTS INC. (US) 2016-06-02 US disclosed
US-9334351-B2 4- and 5-substituted 1,2,3-triazole, and regioisomer mixtures thereof, modified polymers ISP INVESTMENTS INC. (US) 2016-05-10 US disclosed
US-9334351-B2 4- and 5-substituted 1,2,3-triazole, and regioisomer mixtures thereof, modified polymers ISP INVESTMENTS INC. (US) 2016-05-10 US disclosed
US-8993698-B2 4- and 5 substituted 1,2,3-triazole moieties with at least one remote polymerizable moiety and polymers thereof ISP INVESTMENTS INC. (US) 2015-03-31 US disclosed
US-8993698-B2 4- and 5 substituted 1,2,3-triazole moieties with at least one remote polymerizable moiety and polymers thereof ISP INVESTMENTS INC. (US) 2015-03-31 US disclosed
US-20140128550-A1 4- AND 5-SUBSTITUTED 1,2,3-TRIAZOLE, AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS ISP INVESTMENTS INC. (US) 2014-05-08 US disclosed
US-20140128550-A1 4- AND 5-SUBSTITUTED 1,2,3-TRIAZOLE, AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS ISP INVESTMENTS INC. (US) 2014-05-08 US disclosed
WO-2012174400-A1 4-AND 5-SUBSTITUTED 1,2,3-TRIAZOLE AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS ISP INVESTMENTS INC. (US) 2012-12-20 WO disclosed
US-20120142846-A1 4- AND 5 SUBSTITUTED 1,2,3-TRIAZOLE MOIETIES WITH AT LEAST ONE REMOTE POLYMERIZABLE MOIETY AND POLYMERS THEREOF AVOCA LLC 2012-06-07 US disclosed
US-20120142846-A1 4- AND 5 SUBSTITUTED 1,2,3-TRIAZOLE MOIETIES WITH AT LEAST ONE REMOTE POLYMERIZABLE MOIETY AND POLYMERS THEREOF AVOCA LLC 2012-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160152814-A1 4- AND 5-SUBSTITUTED 1,2,3-TRIAZOLE, AND REGIOISOMER MIXTURES THEREOF, MODIFIED POLYMERS MGAT3, MYOC, MLEC HTR1A 2391/4885CYP2D6 1080/4885CYP19A1 2794/4885
US-20120142846-A1 4- AND 5 SUBSTITUTED 1,2,3-TRIAZOLE MOIETIES WITH AT LEAST ONE REMOTE POLYMERIZABLE MOIETY AND POLYMERS THEREOF H1-4, NPY4R, RXFP4 HTR1A 860/4885CYP2D6 2615/4885CYP19A1 1948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.