SCHEMBL10093458

SCHEMBL10093458

COC(=O)c1cncc(-c2cccc(C)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.59
CYP11B1 P15538 3/20 0.59
CYP11B2 P19099 3/20 0.59
CYP2A6 P11509 1/20 0.53
GABRG2 P18507 1/20 0.51
GABRB3 P28472 1/20 0.51
GABRA5 P31644 1/20 0.51
GABRA3 P34903 1/20 0.51
CDK8 P49336 1/20 0.50
NEK1 Q96PY6 4/20 0.49
SLC2A1 P11166 1/20 0.49
CYP19A1 P11511 1/20 0.49
ALDH1A1 P00352 1/20 0.47
MAPK14 Q16539 1/20 0.47
PRMT5 O14744 1/20 0.46
WDR77 Q9BQA1 1/20 0.46
AAK1 Q2M2I8 1/20 0.46
HSD17B10 Q99714 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31418026 0.85 CYP11B1 (0.59) ATMCYP11B1CYP11B2CYP2A6GABRG2
SCHEMBL9008962 0.84 CYP11B1 (0.61) ATMCYP11B1CYP11B2CYP2A6GABRG2
SCHEMBL30285148 0.84 CA12 (0.59) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL7719381 0.84 CA12 (0.59) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL4592371 0.84 CYP11B1 (0.58) ATMCYP11B1CYP11B2CYP2A6GABRG2
SCHEMBL6436030 0.84 CYP11B2 (0.58) ATMCYP11B1CYP11B2CYP2A6GABRG2
SCHEMBL3715051 0.84 ATM (0.69) ATMCYP11B1CYP11B2CYP2A6GABRG2
SCHEMBL27266688 0.83 DHODH (0.57) MAPK14AAK1
SCHEMBL3714867 0.82 ALDH1A1 (0.68) ATMCYP11B1CYP11B2CYP2A6NEK1
SCHEMBL31705350 0.82 ALDH1A1 (0.68) ATMCYP11B1CYP11B2CYP2A6NEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367690-B2 Aminopyridine derivatives having aurora a selective inhibitory action VERTEX PHARMACEUTICALS INC. (US) 2013-02-05 US disclosed
US-20120015969-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION BANYU PHARMACEUTICALS CO., LTD. (JP) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015969-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION AURKA, AURKC, AURKB ATM 2231/4885CYP11B1 940/4885CYP11B2 924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.