SCHEMBL10099702

SCHEMBL10099702

COC(=O)c1nc(-c2cccc(OC)c2)cn1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
TP53 P04637 3/20 0.50
GAA P10253 1/20 0.50
ADORA3 P0DMS8 2/20 0.49
ADORA2B P29275 2/20 0.49
ADORA1 P30542 2/20 0.49
ADORA2A P29274 1/20 0.49
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 2/20 0.48
HTT P42858 1/20 0.48
KDM4E B2RXH2 2/20 0.47
WDR5 P61964 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
PLK1 P53350 1/20 0.47
BRD4 O60885 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260602 0.83 ALDH1A1 (0.51) MAPTSMN1; SMN2GAAALDH1A1NPC1
SCHEMBL12582233 0.76 RAB9A (0.48) MAPTSMN1; SMN2ADORA3ALDH1A1NPC1
SCHEMBL14736254 0.76 PDE10A (0.50) MAPTSMN1; SMN2TP53GAAADORA3
SCHEMBL10099711 0.76 PDE10A (0.54) MAPTSMN1; SMN2TP53GAAADORA1
SCHEMBL2030331 0.75 TLR8 (0.46) MAPTSMN1; SMN2TP53GAAALDH1A1
SCHEMBL3298893 0.75 NPC1 (0.75) MAPTSMN1; SMN2TP53GAAADORA3
SCHEMBL14736793 0.75 PDE10A (0.61) MAPTSMN1; SMN2TP53GAAALDH1A1
SCHEMBL10099708 0.73 MAPT (0.60) MAPTSMN1; SMN2TP53ADORA3ADORA2B
SCHEMBL259679 0.73 PDE10A (0.54) MAPTSMN1; SMN2TP53GAAADORA1
SCHEMBL20085562 0.73 MAPT (0.41) MAPTSMN1; SMN2TP53GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007006-A1 TRIAZOLO- AND PYRAZOLOQUINAZOLINE DERIVATIVES AS PDE10A ENZYME INHIBITOR H. LUNDBECK A/S (DK) 2012-01-19 WO disclosed