SCHEMBL10102465

SCHEMBL10102465

CCOC(=O)c1ccc(OCCCCl)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
HSD17B2 P37059 1/20 0.49
THRA P10827 1/20 0.48
THRB P10828 1/20 0.48
TAS1R3 Q7RTX0 3/20 0.47
TAS1R1 Q7RTX1 3/20 0.47
ESR1 P03372 2/20 0.46
ESR2 Q92731 1/20 0.46
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAOA P21397 1/20 0.45
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3480225 0.90 HSD17B2 (0.54) CA12CA1CA2CA7CA9
SCHEMBL9799085 0.87 TDP1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL12493300 0.86 TAS1R3 (0.60) CA12CA1CA2CA7CA9
SCHEMBL6401723 0.86 HSD17B2 (0.61) HSD17B2LMNAKDM4EMEN1KMT2A
SCHEMBL1715159 0.86 THRA (0.48) CA12CA1CA2CA7CA9
SCHEMBL6582142 0.86 MEN1 (0.53) CA12CA1CA2CA7CA9
SCHEMBL5412826 0.83 KDM4E (0.50) THRATHRBHPGDKDM4ETP53
SCHEMBL27532264 0.82 HSD17B2 (0.47) CA12CA1CA2CA7CA9
SCHEMBL12493009 0.82 CYP1A2 (0.56) THRATHRBTAS1R3TAS1R1ESR1
SCHEMBL1259559 0.81 THRA (0.52) THRATHRBTAS1R3TAS1R1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43098-E1 Nitrogenous heterocyclic compounds and process for making nitrogenous heterocyclic compounds and intermediates thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-01-10 US disclosed