SCHEMBL10103354

SCHEMBL10103354

C=C(C)c1cc(-n2nnc3ccccc32)c(OC)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.48
KDM4E B2RXH2 3/20 0.48
LMNA P02545 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
TSHR P16473 1/20 0.48
RECQL P46063 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KCNMA1 Q12791 1/20 0.43
F12 P00748 3/20 0.42
MGAM O43451 1/20 0.42
AMY1A P0DUB6 1/20 0.42
GAA P10253 1/20 0.42
MIF P14174 1/20 0.42
SI P14410 1/20 0.42
MGAM2 Q2M2H8 1/20 0.42
POLB P06746 1/20 0.41
NR1I2 O75469 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24988440 0.81 KCNMA1 (0.45) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL21183124 0.76 KCNMA1 (0.59) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL2095767 0.72 KDM4E (0.59) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL13620481 0.72 SMN1; SMN2 (0.53) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL2092784 0.72 SMN1; SMN2 (0.59) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL25922416 0.70 KCNMA1 (0.46) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL12202056 0.70 GAA (0.47) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL24633510 0.68 KCNMA1 (0.47) SMN1; SMN2KDM4ELMNANPSR1TSHR
SCHEMBL31062981 0.67 HTT (0.38) LMNARAB9A
SCHEMBL29193567 0.67 SMN1; SMN2 (0.47) SMN1; SMN2KDM4ELMNANPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468735-A1 Synthesis of intermediates for preparing anacetrapib and derivates thereof LEK Pharmaceuticals d.d. (SI) 2012-06-27 EP disclosed