SCHEMBL10107137

SCHEMBL10107137

COc1ccc(/C(C)=N/OCc2ccc3nonc3c2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HTT P42858 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
POLB P06746 1/20 0.41
EPHA2 P29317 1/20 0.39
KDR P35968 1/20 0.39
GAA P10253 2/20 0.38
PDE4D Q08499 5/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL659060 0.91 LMNA (0.39) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL14042218 0.91 ALDH1A1 (0.41) LMNAALDH1A1HTTGAARAB9A
SCHEMBL659059 0.91 LMNA (0.39) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL14042372 0.91 PPARG (0.39) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL660491 0.90 LMNA (0.49) LMNAALDH1A1HTTPPARGPPARA
SCHEMBL10107132 0.90 LMNA (0.49) LMNAALDH1A1HTTPPARGPPARA
SCHEMBL661511 0.90 PPARG (0.44) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL10106850 0.90 PPARG (0.44) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL15255534 0.89 LMNA (0.41) LMNAALDH1A1MAPTKDM4EHTT
SCHEMBL15255533 0.89 LMNA (0.41) LMNAALDH1A1MAPTKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8536157-B2 Non-steroidal compounds THE UNIVERSITY OF MELBOURNE (AU) 2013-09-17 US disclosed
US-20120046255-A1 NON-STEROIDAL COMPOUNDS THE UNIVERSITY OF MELBOURNE of ROYAL PARADE PARKVILLE (AU) 2012-02-23 US disclosed
WO-2008124878-A1 NON-STEROIDAL COMPOUNDS CRYPTOPHARMA PTY LTD (AU) 2008-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046255-A1 NON-STEROIDAL COMPOUNDS PTGES2, PTGES, PTGES3 LMNA 2636/4885ALDH1A1 2237/4885MAPT 2433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.