SCHEMBL1010786

SCHEMBL1010786

CSc1cc(F)cc(C2(O)CCN(C(=O)O)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 6/20 0.40
CCR1 P32246 1/20 0.39
MC4R P32245 1/20 0.37
DRD2 P14416 3/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
PKLR P30613 2/20 0.36
OPRM1 P35372 4/20 0.35
OPRK1 P41145 4/20 0.35
OPRL1 P41146 4/20 0.35
OPRD1 P41143 3/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387449 0.85 S1PR2 (0.43) S1PR2CCR1DRD2DRD4DRD3
SCHEMBL14077927 0.83 DRD2 (0.36) DRD2DRD4DRD3OPRM1OPRK1
SCHEMBL1010791 0.83 GPR119 (0.43) S1PR2DRD2OPRK1OPRD1
SCHEMBL5378448 0.82 S1PR2 (0.39) S1PR2CCR1MC4RDRD2DRD4
SCHEMBL23365187 0.80 S1PR2 (0.40) S1PR2CCR1DRD2DRD4DRD3
SCHEMBL5189318 0.80 DRD2 (0.40) DRD2DRD4DRD3OPRL1
SCHEMBL5376329 0.80 ALDH1A1 (0.46) OPRM1OPRK1OPRL1OPRD1
SCHEMBL3384895 0.79 DRD2 (0.47) S1PR2MC4RDRD2DRD4DRD3
SCHEMBL2535627 0.77 S1PR2 (0.39) S1PR2CCR1DRD2DRD4DRD3
SCHEMBL5367535 0.77 S1PR2 (0.57) S1PR2DRD2OPRM1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948606-B1 3, 5-DISUBSTITUTED PHENYL-PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION NSAB AF NEUROSEARCH SWEDEN AB (DK) 2011-01-05 EP disclosed