SCHEMBL1010847

SCHEMBL1010847

CCOC(=O)Cc1cccc(OCOc2ccc(Br)cc2CNCc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HTT P42858 4/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
LMNA P02545 2/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
KDM4E B2RXH2 2/20 0.45
USP28 Q96RU2 2/20 0.44
USP25 Q9UHP3 2/20 0.44
CCR5 P51681 3/20 0.42
MAPK1 P28482 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1061939 0.80 MEN1 (0.53) ALDH1A1HTTSMN1; SMN2LMNAMEN1
SCHEMBL1943673 0.80 KDM4E (0.53) ALDH1A1HTTSMN1; SMN2LMNAMEN1
SCHEMBL2280306 0.77 FFAR1 (0.44)
SCHEMBL3484087 0.76 NAAA (0.42) ALDH1A1MEN1KMT2AKDM4ECCR5
SCHEMBL6259183 0.75 SMN1; SMN2 (0.63) ALDH1A1HTTSMN1; SMN2LMNAMEN1
SCHEMBL1644681 0.74 F10 (0.44) LMNAMEN1KMT2AMAPK1NPSR1
SCHEMBL1644135 0.74 F10 (0.44) ALDH1A1LMNAMEN1KMT2ANPSR1
SCHEMBL8155074 0.74 CCR5 (0.53) ALDH1A1HTTSMN1; SMN2LMNAMEN1
SCHEMBL2278370 0.74 F10 (0.42) SMN1; SMN2LMNAMEN1KMT2AMAPK1
SCHEMBL2278254 0.73 PPARG (0.48) ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268611-A2 AMINOALKYLPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS Amira Pharmaceuticals, Inc. (US) 2011-01-05 EP disclosed
WO-2009145989-A2 AMINOALKYLPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2009-12-03 WO disclosed