SCHEMBL1011218

SCHEMBL1011218

CCOC(=O)NC(=S)Nc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.64
SMN1; SMN2 Q16637 3/20 0.64
EPHX1 P07099 2/20 0.60
GAA P10253 4/20 0.57
HTT P42858 2/20 0.55
LMNA P02545 2/20 0.55
HPGD P15428 3/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
CRHBP P24387 1/20 0.55
CRHR2 Q13324 1/20 0.55
MAPT P10636 4/20 0.54
ALOX12 P18054 2/20 0.54
MAPK1 P28482 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
TP53 P04637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10688602 0.92 SMN1; SMN2 (0.57) ALDH1A1SMN1; SMN2GAAHTTLMNA
SCHEMBL13313846 0.91 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2EPHX1GAAHTT
SCHEMBL10637569 0.88 HPGD (0.62) ALDH1A1SMN1; SMN2EPHX1GAAHTT
SCHEMBL9023375 0.87 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2GAAHTTLMNA
SCHEMBL21597667 0.87 MEN1 (0.57) ALDH1A1SMN1; SMN2GAALMNAMAPT
SCHEMBL6984178 0.86 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2GAAHTTHPGD
Thiophanate SCHEMBL20842 0.85 ALDH1A1 (0.70) ALDH1A1SMN1; SMN2EPHX1LMNAHPGD
Thiophanate SCHEMBL29398343 0.85 ALDH1A1 (0.70) ALDH1A1SMN1; SMN2EPHX1LMNAHPGD
SCHEMBL23727485 0.85 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2GAAHTTLMNA
SCHEMBL23727417 0.84 EPHX1 (0.62) ALDH1A1SMN1; SMN2EPHX1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 107 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230773-A1 Dipropargyloxybenzene compounds and their production SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1987-08-05 EP claimed
EP-0190036-A2 Fungicidal pyridine derivatives SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1986-08-06 EP claimed
EP-0063905-B1 FUNGICIDAL N-PHENYLCARBAMATES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1985-08-14 EP claimed
EP-0100615-A1 Fungicidal anilides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1984-02-15 EP claimed
US-12617785-B2 Pyrrolo[2,3-b]pyridine-3-carboxamide compositions and methods for ameliorating hearing loss THE ROCKEFELLER UNIVERSITY (US) 2026-05-05 US disclosed
EP-4100008-B1 PYRROLO [2,3-B]PYRIDINE-3-CARBOXAMIDE COMPOSITIONS AND METHODS FOR AMELIORATING HEARING LOSS UNIV ROCKEFELLER (US) 2025-04-02 EP disclosed
US-20240343726-A1 PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION THE ROCKEFELLER UNIVERSITY (US) 2024-10-17 US disclosed
EP-4380562-A1 PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION The Rockefeller University (US) 2024-06-12 EP disclosed
US-20230137893-A1 PYRROLO[2,3-b]PYRIDINE-3-CARBOXAMIDE COMPOSITIONS AND METHODS FOR AMELIORATING HEARING LOSS THE ROCKEFELLER UNIVERSITY (US) 2023-05-04 US disclosed
US-20230137893-A1 PYRROLO[2,3-b]PYRIDINE-3-CARBOXAMIDE COMPOSITIONS AND METHODS FOR AMELIORATING HEARING LOSS THE ROCKEFELLER UNIVERSITY (US) 2023-05-04 US disclosed
WO-2023015156-A1 PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION HUDSPETH A JAMES (US) 2023-02-09 WO disclosed
WO-2023015156-A1 PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION HUDSPETH A JAMES (US) 2023-02-09 WO disclosed
CN-1150800-A Alpha-phenylbutenic acid methyl ester BASF AG (DE) 1997-05-28 CN disclosed
CN-1143359-A Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them BASF AG (DE) 1997-02-19 CN disclosed
CN-1121510-A Substituted phenoxymethylphenyl derivatives, their preparation and their use for controlling pests and fungi BASF AG (DE) 1996-05-01 CN disclosed
CN-1120333-A Imino-substituted phenylacetamides, their preparation and fungicides containing them BASF AG (DE) 1996-04-10 CN disclosed
CN-1109873-A Thioimidates, their preparation and their use BASF AKTEINGESELLSCHAFT (DE) 1995-10-11 CN disclosed
CN-1101040-A Diaryl derivatives and their use as crop protection agents BASF AG (DE) 1995-04-05 CN disclosed
US-5232484-A Aqueous acid solution; mineralization; absence of large concentrations of organic solvents, chloride and sulfate THE CONNECTICUT AGRICULTURAL EXPERIMENT STATION (US) 1993-08-03 US disclosed
US-4086360-A Phenyl thiol carbanilide derivatives, method for the preparation thereof and use thereof as fungicide for agriculture NIPPON KAYAKU KABUSHIKI KAISHA (JA) 1978-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240343726-A1 PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION LATS1, LATS2, YAP1 ALDH1A1 3828/4885SMN1; SMN2 2198/4885EPHX1 4364/4885
US-12617785-B2 Pyrrolo[2,3-b]pyridine-3-carboxamide compositions and methods for ameliorating hearing loss YAP1, LATS2, LATS1 ALDH1A1 2546/4885SMN1; SMN2 2879/4885EPHX1 4502/4885
US-20230137893-A1 PYRROLO[2,3-b]PYRIDINE-3-CARBOXAMIDE COMPOSITIONS AND METHODS FOR AMELIORATING HEARING LOSS LATS2, LATS1, YAP1 ALDH1A1 3775/4885SMN1; SMN2 2796/4885EPHX1 4321/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.