SCHEMBL10114972

SCHEMBL10114972

CC(C)NS(=O)(=O)c1ccc(NC(=O)C2CCC(NS(=O)(=O)C(C)C)CC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.56
LMNA P02545 2/20 0.51
KMT2A Q03164 4/20 0.50
MEN1 O00255 2/20 0.50
USP30 Q70CQ3 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
NAMPT P43490 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14424384 1.00 POLB (0.56) POLBLMNAKMT2AMEN1USP30
SCHEMBL10114911 0.90 KMT2A (0.58) POLBLMNAKMT2AMEN1ALDH1A1
SCHEMBL14424378 0.90 KMT2A (0.58) POLBLMNAKMT2AMEN1ALDH1A1
SCHEMBL10114929 0.87 LMNA (0.56) POLBLMNAKMT2AALDH1A1NPSR1
SCHEMBL13204411 0.87 LMNA (0.56) POLBLMNAKMT2AALDH1A1NPSR1
SCHEMBL13204426 0.87 PTPN1 (0.56) LMNAKMT2AMEN1NPSR1NAMPT
SCHEMBL10114938 0.87 PTPN1 (0.56) LMNAKMT2AMEN1NPSR1NAMPT
SCHEMBL10114584 0.86 LMNA (0.55) POLBLMNAKMT2AMEN1USP30
SCHEMBL14424258 0.86 LMNA (0.55) POLBLMNAKMT2AMEN1USP30
SCHEMBL10114838 0.86 RXFP1 (0.62) KMT2AMEN1RXFP1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8115027-B2 NPY Y5 antagonist SHIONOGI & CO., LTD. (JP) 2012-02-14 US disclosed
US-20100292500-A1 NPY Y5 ANTAGONIST KAWANISHI YASUYUKI 2010-11-18 US disclosed
US-7781461-B2 NPY Y5 antagonist KAWANISHI YASUYUKI 2010-08-24 US disclosed
US-7265130-B2 NPY Y5 antagonist SHIONOGI & CO., LTD. (JP) 2007-09-04 US disclosed
US-20070015762-A1 NPY Y5 antagonist KAWANISHI YASUYUKI 2007-01-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070015762-A1 NPY Y5 antagonist NPY5R, NPY1R, NPY2R POLB 4727/4885LMNA 1925/4885KMT2A 2912/4885
US-20100292500-A1 NPY Y5 ANTAGONIST NPY5R, NPY1R, NPY2R POLB 4751/4885LMNA 2068/4885KMT2A 2768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.