SCHEMBL10117875

SCHEMBL10117875

COC(=O)N(C(=O)OC)c1ncc(-c2ccc(Br)cc2)n1C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NR1H2 P55055 8/20 0.35
DHFR P00374 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
AAK1 Q2M2I8 1/20 0.34
TTK P33981 1/20 0.34
GPR119 Q8TDV5 2/20 0.33
BCL2 P10415 1/20 0.33
IDO1 P14902 1/20 0.33
NR1H3 Q13133 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10117698 0.88 IDO1 (0.41) NPC1RAB9ANR1H2MEN1KMT2A
SCHEMBL10117696 0.86 NR1H2 (0.37) NPC1RAB9ANR1H2MEN1KMT2A
SCHEMBL24176651 0.81 NR1H2 (0.38) NR1H2AAK1TTKGPR119NR1H3
SCHEMBL10117534 0.78 NR1H2 (0.40) NR1H2DHFREGFRERBB2MEN1
SCHEMBL13663132 0.77 PTPN1 (0.53) NPC1RAB9AMEN1KMT2A
SCHEMBL13655217 0.76 NR1H2 (0.35) NR1H2AAK1TTKGPR119NR1H3
SCHEMBL24176882 0.75 CFTR (0.38) NR1H2EGFRTTK
SCHEMBL13655220 0.74 HDAC8 (0.43) SMN1; SMN2NR1H2MEN1KMT2AAAK1
SCHEMBL10117510 0.74 MEN1 (0.45) NPC1RAB9ASMN1; SMN2NR1H2DHFR
SCHEMBL24176646 0.74 HDAC2 (0.35) NPC1RAB9ASMN1; SMN2NR1H2AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed