SCHEMBL10119871

SCHEMBL10119871

Fc1ccc2[nH]cc(CNCC3CCNCC3)c2c1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.72
MAPK1 P28482 1/20 0.53
GPR84 Q9NQS5 1/20 0.51
MPO P05164 10/20 0.50
ALKBH5 Q6P6C2 2/20 0.50
FTO Q9C0B1 2/20 0.50
TSHR P16473 1/20 0.48
HTR2A P28223 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
BRD3 Q15059 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8271475 0.85 SLC6A4 (0.67) SLC6A4GPR84HTR2ATRPM8
SCHEMBL10119820 0.85 SLC6A4 (0.72) SLC6A4GPR84HTR2ATRPM8
SCHEMBL10119730 0.85 SLC6A4 (0.51) SLC6A4FTOHTR2A
SCHEMBL5726056 0.84 SLC6A4 (1.00) SLC6A4MAPK1GPR84MPOTSHR
SCHEMBL10119656 0.82 SLC6A4 (0.69) SLC6A4GPR84
SCHEMBL9635299 0.81 SLC6A4 (0.78) SLC6A4MAPK1GPR84MPOHTR2A
SCHEMBL1970036 0.80 MPO (0.70) SLC6A4MPOHTR2ATRPM8
SCHEMBL8125191 0.79 SLC6A4 (0.84) SLC6A4MAPK1GPR84MPOTSHR
Succinic Acid SCHEMBL6794738 0.78 SLC6A4 (0.81) SLC6A4MAPK1GPR84MPOTSHR
SCHEMBL2805245 0.76 GPR84 (0.59) SLC6A4MAPK1GPR84MPOTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781639-B1 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE JANSSEN PHARMACEUTICA NV (BE) 2012-01-25 EP disclosed