SCHEMBL10120997

SCHEMBL10120997

C=C1N[C@](CCC2CCCCC2)(C[C@H]2CCC[C@@H](Nc3ccccc3)C2)C(=O)N1C

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.49
CTSD P07339 14/20 0.49
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
HPGD P15428 1/20 0.35
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7538302 0.89 BACE1 (0.51) BACE1CTSDPRMT5WDR77HPGD
SCHEMBL7531658 0.89 BACE1 (0.51) BACE1CTSDPRMT5WDR77HPGD
SCHEMBL7533881 0.89 BACE1 (0.51) BACE1CTSDPRMT5WDR77HPGD
SCHEMBL10121022 0.87 BACE1 (0.45) BACE1CTSDPRMT5WDR77HPGD
SCHEMBL10121026 0.85 BACE1 (0.50) BACE1CTSD
SCHEMBL10121006 0.82 BACE1 (0.44) BACE1CTSDPRMT5WDR77
SCHEMBL10121004 0.81 BACE1 (0.46) BACE1CTSD
SCHEMBL10121023 0.81 BACE1 (0.47) BACE1CTSD
SCHEMBL10121024 0.81 BACE1 (0.47) BACE1CTSD
SCHEMBL10121020 0.80 KDM4E (0.44) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178513-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-15 US disclosed