SCHEMBL10121022

SCHEMBL10121022

C=C1N[C@](CCC2CCCCC2)(C[C@H]2CCCC(Nc3ccccn3)C2)C(=O)N1C

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.45
CTSD P07339 14/20 0.45
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7538345 0.90 BACE1 (0.46) BACE1CTSDMEN1HPGDKMT2A
SCHEMBL7537566 0.90 BACE1 (0.46) BACE1CTSDMEN1HPGDKMT2A
SCHEMBL10120997 0.87 BACE1 (0.49) BACE1CTSDHPGDPRMT5WDR77
SCHEMBL10121023 0.81 BACE1 (0.47) BACE1CTSD
SCHEMBL10121024 0.81 BACE1 (0.47) BACE1CTSD
SCHEMBL10121020 0.80 KDM4E (0.44) BACE1CTSD
SCHEMBL8198551 0.80 BACE1 (0.43) BACE1CTSDHPGD
SCHEMBL13054411 0.80 BACE1 (0.43) BACE1CTSDHPGD
SCHEMBL2965484 0.80 BACE1 (0.43) BACE1CTSDHPGD
SCHEMBL2965482 0.80 BACE1 (0.43) BACE1CTSDHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178513-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-15 US disclosed