SCHEMBL10123568

SCHEMBL10123568

C=C(NNc1ccccc1Cl)NC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 4/20 0.44
PDK2 Q15119 4/20 0.44
PDK3 Q15120 4/20 0.44
PDK4 Q16654 4/20 0.44
MAPT P10636 4/20 0.41
HTT P42858 2/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CRHR1 P34998 5/20 0.39
P2RX7 Q99572 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
NPC1 O15118 1/20 0.35
GLA P06280 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10123569 0.78 ALDH1A1 (0.45) PDK1PDK2PDK3PDK4MAPT
SCHEMBL10123574 0.73 GAA (0.40) PDK1PDK2PDK3PDK4MAPT
SCHEMBL10123576 0.73 GAA (0.34) MAPTHTTGAALMNAKMT2A
SCHEMBL10122312 0.73 MAPT (0.70) PDK1PDK2PDK3PDK4MAPT
SCHEMBL10123535 0.72 ABCB1 (0.35) MAPTHTTGAALMNAALDH1A1
SCHEMBL10123572 0.70 KDM4E (0.42) MAPTHTTGAALMNAALDH1A1
SCHEMBL10123578 0.70 GAA (0.42) PDK1PDK2PDK3PDK4MAPT
SCHEMBL10123534 0.70 GAA (0.43) MAPTHTTGAAALDH1A1MEN1
SCHEMBL10123461 0.69 MEN1 (0.38) MAPTHTTGAALMNAALDH1A1
SCHEMBL5211507 0.68 MEN1 (0.61) PDK1PDK2PDK3PDK4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012060820-A1 SULFONYL SEMICARBAZIDES, SEMICARBAZIDES AND UREAS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS FOR TREATING HEMORRHAGIC FEVER VIRUSES, INCLUDING INFECTIONS ASSOCIATED WITH ARENAVIRUSES SIGA TECHNOLOGIES, INC. (US) 2012-05-10 WO disclosed