SCHEMBL10123576

SCHEMBL10123576

C=C(NNc1cccc2c(N(C)C)cccc12)NC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.34
HTT P42858 2/20 0.34
MAPT P10636 2/20 0.34
CA2 P00918 1/20 0.34
LMNA P02545 1/20 0.34
F2 P00734 3/20 0.33
PRSS1 P07477 3/20 0.33
PRSS2 P07478 3/20 0.33
PRSS3 P35030 3/20 0.33
MCL1 Q07820 1/20 0.32
CHEK1 O14757 1/20 0.32
NEK2 P51955 1/20 0.32
LIMK1 P53667 1/20 0.32
DYRK1A Q13627 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
EDNRA P25101 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10123568 0.73 PDK1 (0.44) GAAHTTMAPTLMNAL3MBTL1
SCHEMBL10123569 0.69 ALDH1A1 (0.45) GAAHTTMAPTLMNAF2
SCHEMBL10123535 0.69 ABCB1 (0.35) GAAHTTMAPTLMNAKDM4E
SCHEMBL10122106 0.68 F2 (0.49) CA2F2PRSS1PRSS2PRSS3
SCHEMBL10123534 0.67 GAA (0.43) GAAHTTMAPTL3MBTL1KMT2A
SCHEMBL10123461 0.66 MEN1 (0.38) GAAHTTMAPTLMNAL3MBTL1
SCHEMBL27372318 0.65 CA2 (0.50) HTTCA2F2PRSS1PRSS2
SCHEMBL10123578 0.64 GAA (0.42) GAAHTTMAPTLMNAL3MBTL1
SCHEMBL14920003 0.64 CA2 (0.42) GAAHTTCA2F2PRSS1
SCHEMBL14920002 0.64 CA2 (0.50) HTTCA2F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012060820-A1 SULFONYL SEMICARBAZIDES, SEMICARBAZIDES AND UREAS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS FOR TREATING HEMORRHAGIC FEVER VIRUSES, INCLUDING INFECTIONS ASSOCIATED WITH ARENAVIRUSES SIGA TECHNOLOGIES, INC. (US) 2012-05-10 WO disclosed
WO-2008147474-A2 SULFONYL SEMICARBAZIDES, CARBONYL SEMICARBAZIDES, SEMICARBAZIDES AND UREAS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS FOR TREATING HEMORRHAGIC FEVER VIRUSES, INCLUDING INFECTIONS ASSOCIATED WITH ARENAVIRUSES SIGA TECHNOLOGIES, INC. (US) 2008-12-04 WO disclosed