SCHEMBL10123535

SCHEMBL10123535

C=C(NNc1cccc2c1OCCO2)NC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.35
FLT1 P17948 1/20 0.35
MTNR1A P48039 10/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
MRGPRX1 Q96LB2 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ACLY P53396 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10123568 0.72 PDK1 (0.44) LMNAGAAMAPTHTTKDM4E
SCHEMBL10123576 0.69 GAA (0.34) LMNAGAAMAPTHTTKDM4E
SCHEMBL10123569 0.68 ALDH1A1 (0.45) LMNAGAAMAPTHTTKDM4E
SCHEMBL10122196 0.68 ACLY (0.41) MTNR1ALMNAGAAMAPTHTT
SCHEMBL10123534 0.66 GAA (0.43) GAAMAPTHTTKDM4EALDH1A1
SCHEMBL8306057 0.66 MTNR1A (0.45) ABCB1FLT1MTNR1ALMNAHTT
SCHEMBL7431136 0.65 MRGPRX1 (0.48) ABCB1FLT1MTNR1ALMNAMAPT
SCHEMBL10123461 0.65 MEN1 (0.38) LMNAGAAMAPTHTTKDM4E
Hydrochloric Acid SCHEMBL2461132 0.64 MTNR1A (0.44) MTNR1ALMNAHTTMRGPRX1KDM4E
SCHEMBL10123578 0.64 GAA (0.42) LMNAGAAMAPTHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012060820-A1 SULFONYL SEMICARBAZIDES, SEMICARBAZIDES AND UREAS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS FOR TREATING HEMORRHAGIC FEVER VIRUSES, INCLUDING INFECTIONS ASSOCIATED WITH ARENAVIRUSES SIGA TECHNOLOGIES, INC. (US) 2012-05-10 WO disclosed