SCHEMBL10124052

SCHEMBL10124052

O=C1CCCc2c1cnn2-c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.67
CA4 P22748 10/20 0.67
CA2 P00918 9/20 0.67
CA9 Q16790 8/20 0.67
HTT P42858 1/20 0.52
PLK1 P53350 1/20 0.51
CSNK2A1 P68400 1/20 0.51
PLK3 Q9H4B4 1/20 0.51
GPR52 Q9Y2T5 1/20 0.45
ELANE P08246 2/20 0.44
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10124062 0.91 CA1 (0.55) CA1CA4CA2CA9HTT
SCHEMBL19031814 0.85 CA1 (0.72) CA1CA4CA2CA9HTT
SCHEMBL2512530 0.84 CA1 (0.67) CA1CA4CA2CA9HTT
SCHEMBL3133796 0.81 CA1 (0.63) CA1CA4CA2CA9HTT
SCHEMBL12294731 0.81 CA1 (0.58) CA1CA4CA2CA9HTT
SCHEMBL14985286 0.80 HTT (0.51) CA1CA4CA2CA9HTT
SCHEMBL17583960 0.80 CA1 (0.64) CA1CA4CA2CA9HTT
SCHEMBL958124 0.78 CA1 (0.59) CA1CA4CA2CA9HTT
SCHEMBL18825197 0.77 CA1 (0.50) CA1CA4CA2CA9HTT
SCHEMBL19031800 0.75 CA1 (0.65) CA1CA4CA2CA9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016961-B1 NOVEL RUTHENIUM CATALYSTS AND THEIR USE FOR ASYMMETRIC REDUCTION OF KETONES BOEHRINGER INGELHEIM INT (DE) 2017-11-15 EP disclosed
US-9029540-B2 Ruthenium catalysts and their use for asymmetric reduction of ketones BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-05-12 US disclosed
US-9029540-B2 Ruthenium catalysts and their use for asymmetric reduction of ketones BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-05-12 US disclosed
EP-2655371-B1 PYRAZOLOPIPERIDINE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2015-02-25 EP disclosed
WO-2015002769-A1 NOVEL RUTHENIUM CATALYSTS AND THEIR USE FOR ASYMMETRIC REDUCTION OF KETONES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-01-08 WO disclosed
US-20150005500-A1 NOVEL RUTHENIUM CATALYSTS AND THEIR USE FOR ASYMMETRIC REDUCTION OF KETONES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-01-01 US disclosed
US-20150005500-A1 NOVEL RUTHENIUM CATALYSTS AND THEIR USE FOR ASYMMETRIC REDUCTION OF KETONES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-01-01 US disclosed
US-8546442-B2 Pyrazolopiperidine compounds as CCR1 receptor antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-10-01 US disclosed
US-8546442-B2 Pyrazolopiperidine compounds as CCR1 receptor antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-10-01 US disclosed
US-20120322790-A1 Pyrazolopiperidine Compounds As CCR1 Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-20 US disclosed
US-20120322790-A1 Pyrazolopiperidine Compounds As CCR1 Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-20 US disclosed
WO-2012087782-A1 PYRAZOLOPIPERIDINE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120322790-A1 Pyrazolopiperidine Compounds As CCR1 Receptor Antagonists CCR1, CCR3, CCR4 CA1 2076/4885CA4 3405/4885CA2 3581/4885
US-20150005500-A1 NOVEL RUTHENIUM CATALYSTS AND THEIR USE FOR ASYMMETRIC REDUCTION OF KETONES PDHB, CYP2E1, PDK1 CA1 2004/4885CA4 2749/4885CA2 3967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.