SCHEMBL10125435

SCHEMBL10125435

N#CC1(c2ccc(C(F)(F)F)cc2CCc2ccnc(Nc3ccc(N)c(CC=O)c3)n2)CCC1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 2/20 0.33
KCNH2 Q12809 1/20 0.32
SCN9A Q15858 1/20 0.32
AURKA O14965 8/20 0.32
MET P08581 1/20 0.31
KDR P35968 1/20 0.31
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669800 0.81 PTK2B (0.46) AURKAMETKDR
SCHEMBL10125436 0.75 MAP3K12 (0.36) MAP3K12
SCHEMBL15023735 0.75 PTK2B (0.46)
SCHEMBL10125761 0.70 TBK1 (0.45) MET
SCHEMBL10125381 0.66 PTK2B (0.47)
SCHEMBL10125382 0.66 TBK1 (0.45) MET
SCHEMBL15023744 0.65 PTK2B (0.49)
SCHEMBL669843 0.65 PTK2B (0.49)
SCHEMBL10125760 0.64 PTK2B (0.51) AURKAMETKDR
SCHEMBL10125762 0.64 PTK2B (0.51) AURKAMETKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012022408-A1 PYRIMIDINE DERIVATIVES AS FAK INHIBITORS MERCK PATENT GMBH (DE) 2012-02-23 WO disclosed