SCHEMBL10129665

SCHEMBL10129665

C[C@H]1Oc2ccc(N3C(=O)c4ccccc4C3=O)cc2N(C)C1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.47
MEN1 O00255 3/20 0.47
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
ABCC8 Q09428 1/20 0.41
KCNJ11 Q14654 1/20 0.41
TSHR P16473 1/20 0.40
GRM4 Q14833 1/20 0.40
MAOA P21397 1/20 0.40
PIM3 Q86V86 1/20 0.39
HIPK4 Q8NE63 1/20 0.39
SCN2A Q99250 1/20 0.39
CA9 Q16790 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10129676 1.00 KMT2A (0.47) KMT2AMEN1PDE3BPDE3AABCC8
SCHEMBL10151420 0.77 MEN1 (0.48) KMT2AMEN1PDE3BPDE3AGRM4
SCHEMBL10130351 0.75 TSHR (0.58) KMT2AMEN1PDE3BPDE3AABCC8
SCHEMBL10129864 0.75 TSHR (0.58) KMT2AMEN1PDE3BPDE3AABCC8
SCHEMBL10130347 0.75 TSHR (0.58) KMT2AMEN1PDE3BPDE3AABCC8
SCHEMBL10129660 0.75 PARP1 (0.56) KMT2AMEN1PDE3BPDE3APIM3
SCHEMBL10129675 0.75 PARP1 (0.56) KMT2AMEN1PDE3BPDE3APIM3
SCHEMBL3401752 0.74 TSHR (0.51) KMT2AMEN1PDE3BPDE3ATSHR
SCHEMBL29354025 0.74 TSHR (0.51) KMT2AMEN1PDE3BPDE3ATSHR
SCHEMBL10129667 0.74 PDE3B (0.50) KMT2AMEN1PDE3BPDE3AABCC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106190-B2 2-aminobenzamide derivatives ASTELLAS PHARMA INC. (JP) 2012-01-31 US disclosed
US-8106190-B2 2-aminobenzamide derivatives ASTELLAS PHARMA INC. (JP) 2012-01-31 US disclosed
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2009-09-17 US disclosed
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE TRPV1, TRPV2, TRPV5 KMT2A 2104/4885MEN1 3066/4885PDE3B 1598/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.