SCHEMBL10130332

SCHEMBL10130332

CCc1cccc(N(C)N)c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.53
TP53 P04637 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
THPO P40225 1/20 0.46
MTOR P42345 1/20 0.46
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
PMP22 Q01453 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18469383 0.83 SIGMAR1 (0.49) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL17485887 0.83 SIGMAR1 (0.51) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL129446 0.83 SIGMAR1 (0.51) SIGMAR1TSHRKMT2A
SCHEMBL30966769 0.83 SIGMAR1 (0.51) SIGMAR1TSHRKMT2A
SCHEMBL4487876 0.82 SIGMAR1 (0.47) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7258873 0.82 NOS1 (0.50) SIGMAR1TSHR
Hydrochloric Acid SCHEMBL2867283 0.81 SIGMAR1 (0.53) SIGMAR1TSHRMEN1LMNAMAPT
SCHEMBL25922215 0.81 SIGMAR1 (0.50) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL18499750 0.79 SIGMAR1 (0.53) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7263645 0.79 TAAR1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212287-B1 PIPERIDINYL AND PIPERAZINYL MODULATORS OF y-SECRETASE JANSSEN PHARMACEUTICA NV (BE) 2012-02-01 EP disclosed
US-4092308-A 4-Sulphomethyl substituted hydroxypyridone azo dyestuffs CIBA-GEIGY CORPORATION (US) 1978-05-30 US disclosed