SCHEMBL10137757

SCHEMBL10137757

CC(Cc1ccccc1)C(O)C#N

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.56
CYP2D6 P10635 1/20 0.52
MAOB P27338 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TAAR1 Q96RJ0 4/20 0.45
SLC6A2 P23975 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
SLC18A2 Q05940 1/20 0.42
CTSC P53634 3/20 0.41
ANPEP P15144 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13534723 1.00 TRPA1 (0.56) TRPA1CYP2D6MAOBNPC1RAB9A
SCHEMBL933101 0.81 TRPA1 (0.56) TRPA1CYP2D6MAOBTAAR1SLC6A2
SCHEMBL21852752 0.79 TRPA1 (0.69) TRPA1CYP2D6NPC1RAB9ATAAR1
SCHEMBL234669 0.79 TRPA1 (0.69) TRPA1CYP2D6NPC1RAB9ATAAR1
SCHEMBL19725385 0.79 TRPA1 (0.69) TRPA1CYP2D6NPC1RAB9ATAAR1
Water SCHEMBL3896311 0.79 TRPA1 (0.74) TRPA1CYP2D6MAOBTAAR1SLC6A2
SCHEMBL4951816 0.77 TRPA1 (0.67) TRPA1CYP2D6NPC1RAB9ATAAR1
SCHEMBL11412673 0.77 EPHX1 (0.48) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8690443 0.77 EPHX1 (0.48) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL27313237 0.77 CYP2D6 (0.62) TRPA1CYP2D6MAOBTAAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43298-E1 Peptides as NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2012-04-03 US disclosed
US-20110117057-A1 NOVEL PEPTIDES AS NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2011-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110117057-A1 NOVEL PEPTIDES AS NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS HPN, TMPRSS15, VIP TRPA1 3380/4885CYP2D6 3181/4885MAOB 3346/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.